What it is: InstaMed's BPC-157 Sublingual Oral Strip delivers 500 mcg of high-purity BPC-157 per strip in a needle-free, sublingual dissolving format using proprietary InstaRelease® delivery technology — the buccal membrane transmucosal absorption system that bypasses first-pass hepatic metabolism for direct systemic peptide delivery. BPC-157 (Body Protection Compound-157) is a 15-amino acid synthetic peptide sequence originally identified within human gastric juice proteins, with an extensive preclinical research profile spanning tissue repair, tendon and ligament regeneration, gut mucosal integrity, vascular angiogenesis, and neuroprotection. Each strip is third-party CoA-verified at 98.8% purity by HPLC. Exclusively practitioner-directed.
How it works: BPC-157 supports tissue repair and regenerative signaling through multiple convergent mechanisms. It upregulates growth hormone receptor expression in tendon fibroblasts, accelerating tendon-to-bone healing and collagen matrix reorganization. It promotes angiogenesis through VEGF pathway activation — supporting vascular tissue repair and the neovascularization required for musculoskeletal and gastrointestinal tissue regeneration. It modulates nitric oxide synthesis to support vascular tone and blood flow to injured tissue. In the gastrointestinal system, BPC-157 supports mucosal integrity by promoting cytoprotective prostaglandin synthesis and inhibiting cytokine-driven mucosal inflammation. InstaRelease® buccal strip delivery enables transmucosal BPC-157 absorption — bypassing the gastrointestinal degradation that limits conventional oral peptide delivery — with CoA-confirmed Penetratin (a cell-penetrating peptide) at 0.006 mg/strip facilitating mucosal membrane permeation and peptide uptake.
When to use it: Indicated for adults in practitioner-directed protocols requiring tissue repair support — including tendon, ligament, and muscle recovery, gastrointestinal mucosal integrity support, vascular health, and cellular regeneration. One strip sublingually 5 days per week with 2 days off. Optimal protocol duration is 8–12 weeks. Not recommended during pregnancy or breastfeeding. Consult a healthcare practitioner before use if managing a medical condition or taking medications.
Serving Size: 1 Strip
Servings Per Container: 20
Suggested Use: Place one strip on the tongue and allow it to dissolve, then swallow. Take 1 strip daily, 5 days per week with 2 days off. An 8–12 week cycle is optimal, or as directed by your healthcare practitioner.
| Ingredient | Amount Per Serving | % Daily Value |
|---|---|---|
| Calories | 0 | — |
| Calories from Fat | 0 | — |
| Total Fat | 0 | 0% |
| BPC-157 | 500 mcg | † |
† Daily Value not established.
Other Ingredients: Pullulan, β-cyclodextrin, stevia, vegetable glycerin, organic strawberry flavor extract, xanthan gum, arabic gum, citric acid, sunflower lecithin, beet powder (color).
Caution: Not recommended during pregnancy or breastfeeding. Consult your healthcare practitioner before use if taking any medications or managing a medical condition. For adult use only. Keep out of reach of children. Store in a cool, dry place away from direct sunlight and excessive heat. Do not use if inner seal is broken or missing.
✓ Gluten Free ✓ Soy Free ✓ Non-GMO ✓ Needle-Free ✓ Third-Party CoA Verified ✓ No Artificial Colors or Flavors
Key Ingredients:
BPC-157 (Body Protection Compound-157) — 500 mcg BPC-157 is a 15-amino acid synthetic peptide sequence (Gly-Glu-Pro-Pro-Pro-Gly-Lys-Pro-Ala-Asp-Asp-Ala-Gly-Leu-Val) originally identified within the cytoprotective protein fraction of human gastric juice, delivered here at 500 mcg per strip with third-party CoA verification of 98.8% purity by HPLC and full conformance across heavy metals and microbial specifications. BPC-157's primary tissue-repair mechanisms include upregulation of growth hormone receptor expression in tendon fibroblasts to accelerate collagen synthesis and tendon-to-bone healing, VEGF-mediated angiogenesis activation to support neovascularization and blood flow in injured musculoskeletal and gastrointestinal tissues, nitric oxide pathway modulation supporting vascular tone and tissue perfusion, and cytoprotective prostaglandin synthesis promotion in gastrointestinal mucosal cells to support barrier integrity and mucosal healing. Delivered via InstaRelease® buccal strip technology, BPC-157 undergoes transmucosal absorption through the sublingual and buccal mucosa — bypassing the first-pass hepatic metabolism and gastrointestinal peptide degradation that significantly limit conventional oral peptide bioavailability — in a needle-free, pre-dosed, travel-compatible format for practitioner-directed tissue repair and regenerative protocols.
InstaRelease® Delivery Technology (Buccal Transmucosal Strip Matrix) The InstaRelease® oral dissolving strip matrix is InstaMed's proprietary buccal transmucosal delivery platform — engineered from pullulan (a water-soluble polysaccharide film-forming agent), β-cyclodextrin (a cyclic oligosaccharide that forms inclusion complexes with peptides to improve dissolution and mucosal contact), and Penetratin (a cell-penetrating peptide confirmed at 0.006 mg/strip by CoA, facilitating transmucosal membrane permeation and intracellular peptide uptake). This matrix enables direct mucosal absorption of BPC-157 through the buccal and sublingual mucosa — delivering the peptide into systemic circulation without injection, without water, and without the GI degradation that undermines conventional oral peptide formats. The result is a convenient, consistently pre-dosed, high-compliance delivery system that brings clinical-grade peptide administration into everyday practitioner and client use without the barrier of injectable protocols.
